2008JSPC Award for Excellence
1P-03 A Practical Synthesis of the PDE4 inhibitor KW-4490
Arata Yanagisawa*, Koichiro Nishimura ,Tetsuya Nezu, Kyoji Ando, Ayako Maki,
Eiichiro Imai, Shin-ichiro Mohri (Kyowa Hakko Kogyo, Japan)
1P-22 An Efficient Synthesis of the PKCb Inhibitor JTT-010
Using a Novel Cyclopropane Ring-Opening Reaction with Indole
Takashi Inaba*, Masahiro Tanaka, Minoru Ubukata, Takafumi Matsuo, Katsutaka Yasue,
Katsuya Matsumoto, Yasuyuki Kajimoto, Takashi Ogo (Japan Tobacco Inc.,Japan)
1P-31 Development of Protecting Group Free Catalytic O-Selective Acylation of Aminoalcohols
Takashi Ohshima*, Takanori Iwasaki, Yusuke Maegawa, Yukiko Hayashi, Kazushi Mashima (Osaka University, Japan)
2P-73 Dynamic Kinetic Resolution of Primary Amines by Lipase-Palladium Cocatalysis
Kiwon Han*, Yoon Kyung Choi, Cheolwoo Kim, Jaiwook Park, Mahn-Joo Kim (POSTECH, Korea)